SCHEMBL7530107

SCHEMBL7530107

CCC[C@H](NC(=O)C1(NC(=O)c2cc(OC)cc(OC)c2)CCCCC1)C(=O)c1nc2ccccc2o1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.58
CTSS P25774 12/20 0.58
CTSL P07711 11/20 0.58
CTSB P07858 11/20 0.58
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 2/20 0.42
KMT2A Q03164 2/20 0.42
HSD17B10 Q99714 2/20 0.42
USP2 O75604 1/20 0.42
GAA P10253 1/20 0.42
STAT3 P40763 1/20 0.42
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
NPPA P01160 2/20 0.40
MME P08473 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7530008 0.93 CTSK (0.63) CTSKCTSSCTSLCTSBKDM4E
SCHEMBL7528076 0.89 CTSL (0.54) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL7531164 0.87 CTSS (0.54) CTSKCTSSCTSLCTSBNPPA
SCHEMBL7533061 0.86 CTSS (0.56) CTSKCTSSCTSLCTSBNPPA
SCHEMBL7530187 0.86 CTSS (0.57) CTSKCTSSCTSLCTSBNPPA
SCHEMBL7526705 0.85 CTSS (0.55) CTSKCTSSCTSLCTSBNPPA
SCHEMBL7532290 0.85 CTSS (0.58) CTSKCTSSCTSLCTSBHPGD
SCHEMBL7528445 0.85 CTSS (0.74) CTSKCTSSCTSLCTSBNPPA
SCHEMBL7531445 0.85 CTSS (0.49) CTSKCTSSCTSLCTSBNPPA
SCHEMBL7530137 0.85 CTSS (0.62) CTSKCTSSCTSLCTSBNPPA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002023784-A2 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-03-21 WO claimed
WO-2002023784-A2 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-03-21 WO disclosed