SCHEMBL7530169

SCHEMBL7530169

c1ccc(CCN2CCC3=C(CCc4ccccc43)C2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.97
PARP1 P09874 1/20 0.54
DRD2 P14416 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9309721 0.83 SIGMAR1 (0.97) SIGMAR1PARP1
SCHEMBL9309563 0.81 SIGMAR1 (0.97) SIGMAR1PARP1
Hydrochloric Acid SCHEMBL9308175 0.80 SIGMAR1 (1.00) SIGMAR1PARP1
SCHEMBL6512477 0.76 HRH3 (0.68) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9306818 0.74 SIGMAR1 (0.64) SIGMAR1
SCHEMBL7378750 0.73 SLC6A3 (0.58) SIGMAR1DRD2
Hydrochloric Acid SCHEMBL9308470 0.73 SIGMAR1 (0.67) SIGMAR1
SCHEMBL7386396 0.73 SIGMAR1 (1.00) SIGMAR1PARP1
SCHEMBL10565610 0.72 HTR1A (0.71) SIGMAR1PARP1DRD2HTR2A
SCHEMBL31629019 0.72 SLC6A3 (0.56) SIGMAR1DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002030422-A1 USE OF DEFINED SUBSTANCES THAT BIND TO THE SIGMA RECEPTOR FOR COMBATING SARCOMA AND CARCINOMA MERCK PATENT GMBH (DE) 2002-04-18 WO claimed
WO-2002030422-A1 USE OF DEFINED SUBSTANCES THAT BIND TO THE SIGMA RECEPTOR FOR COMBATING SARCOMA AND CARCINOMA MERCK PATENT GMBH (DE) 2002-04-18 WO disclosed
WO-2002030422-A1 USE OF DEFINED SUBSTANCES THAT BIND TO THE SIGMA RECEPTOR FOR COMBATING SARCOMA AND CARCINOMA MERCK PATENT GMBH (DE) 2002-04-18 WO disclosed