SCHEMBL7531476

SCHEMBL7531476

Cc1cc(Br)cc(C)c1NC=O

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
RAPGEF4 Q8WZA2 3/20 0.35
DHFR P00374 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14858457 0.82 ERN1 (0.45) ALDH1A1MAPTHPGD
SCHEMBL2093540 0.81 RAPGEF4 (0.52) ALDH1A1RAPGEF4
SCHEMBL11915499 0.77 ALDH1A1 (0.39) ALDH1A1HTR1DHTR1BTAS1R3TAS1R1
SCHEMBL8716465 0.77 CYP3A4 (0.46) ALDH1A1MAPTHPGDRAPGEF4
SCHEMBL10501503 0.77 ALDH1A1 (0.36) ALDH1A1RAPGEF4
SCHEMBL16520251 0.77 HMGB1 (0.38) ALDH1A1RAPGEF4
SCHEMBL10500612 0.74 FFAR4 (0.47) ALDH1A1HPGDRAPGEF4
SCHEMBL10499823 0.74 TSHR (0.35) ALDH1A1MAPTRAPGEF4
SCHEMBL25732352 0.74 LMNA (0.35) RAPGEF4
SCHEMBL25732294 0.74 S1PR4 (0.35) ALDH1A1MAPTRAPGEF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed