SCHEMBL7533150

SCHEMBL7533150

c1ccc(Cc2cscn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.48
SLC6A3 Q01959 6/20 0.47
CALM1 P0DP23 1/20 0.44
GPR142 Q7Z601 2/20 0.43
ALDH1A1 P00352 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 1/20 0.41
GRM5 P41594 1/20 0.40
NPC1 O15118 1/20 0.40
AOC3 Q16853 1/20 0.39
FYN P06241 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6286235 0.84 LTA4H (0.44) LTA4HSLC6A3GPR142ALDH1A1RAB9A
Eprodisate SCHEMBL27535860 0.83 LTA4H (0.42) LTA4HSLC6A3GPR142RAB9ASMN1; SMN2
SCHEMBL29991111 0.78 FYN (0.46) LTA4HSLC6A3FYN
SCHEMBL7992030 0.77 GPR142 (0.49) SLC6A3GPR142TDP1
SCHEMBL29131248 0.77 NPC1 (0.46) SLC6A3GPR142ALDH1A1RAB9ASMN1; SMN2
SCHEMBL7493474 0.75 SLC6A4 (0.41) LTA4HSLC6A3GPR142ALDH1A1RAB9A
SCHEMBL29131241 0.74 SLC6A3 (0.41) SLC6A3GPR142RAB9ASMN1; SMN2SLC6A2
SCHEMBL29131243 0.74 SLC6A3 (0.41) SLC6A3GPR142RAB9ASMN1; SMN2SLC6A2
SCHEMBL6031397 0.73 GAA (0.53) GPR142SMN1; SMN2
SCHEMBL6001756 0.73 SLC6A3 (0.41) SLC6A3RAB9ASMN1; SMN2L3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101980706-A Combination of a dithiazole salt or precursor thereof and artemisinin or a derivative thereof for the treatment of acute malaria SANOFI AVENTIS 2011-02-23 CN claimed
US-12016312-B2 Animal models, screening methods, and treatment methods for intraocular diseases or disorders Smilebiotek Zhuhai Limited (CN) 2024-06-25 US disclosed
CN-101980706-B Combination of salts of Chinese pulsatilla thiazolicola or precursors thereof and artemisinin or derivatives thereof for the treatment of acute malaria SANOFI AVENTIS 2013-11-27 CN disclosed
CN-101980706-A Combination of a dithiazole salt or precursor thereof and artemisinin or a derivative thereof for the treatment of acute malaria SANOFI AVENTIS 2011-02-23 CN disclosed
CN-101528691-A Matrix metalloproteinase inhibitors RANBAXY LAB LTD (IN) 2009-09-09 CN disclosed
EP-1196371-A1 QUATERNARY BIS-AMMONIUM SALT PRECURSORS AND THEIR USES AS PRODRUGS HAVING AN ANTIPARASITIC ACTIVITY CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2002-04-17 EP disclosed
WO-2001005742-A1 QUATERNARY BIS-AMMONIUM SALT PRECURSORS AND THEIR USES AS PRODRUGS HAVING AN ANTIPARASITIC ACTIVITY CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 2001-01-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12016312-B2 Animal models, screening methods, and treatment methods for intraocular diseases or disorders MB, MYOC, PDE6A LTA4H 450/4885SLC6A3 2449/4885CALM1 3826/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.