SCHEMBL7533710

SCHEMBL7533710

O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1sccc1NS(=O)(=O)c1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.70
PTGS1 P23219 1/20 0.70
SCN3A Q9NY46 5/20 0.64
SCN5A Q14524 2/20 0.64
SCN9A Q15858 2/20 0.64
SCN1A P35498 1/20 0.64
SCN4A P35499 1/20 0.64
SCN2A Q99250 1/20 0.64
SCN8A Q9UQD0 1/20 0.64
SCN10A Q9Y5Y9 1/20 0.64
KMT2A Q03164 8/20 0.63
MEN1 O00255 7/20 0.63
ALDH1A1 P00352 3/20 0.63
CA1 P00915 1/20 0.63
PKM P14618 2/20 0.61
RXFP1 Q9HBX9 2/20 0.61
LMNA P02545 1/20 0.60
TSHR P16473 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
MAPK1 P28482 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7531142 0.90 POLB (0.59) CYP3A4PTGS1SCN3ASCN5ASCN9A
SCHEMBL7530791 0.87 POLB (0.56) CYP3A4PTGS1SCN3ASCN5ASCN9A
SCHEMBL7531704 0.85 ALDH1A1 (0.57) CYP3A4PTGS1KMT2AMEN1ALDH1A1
SCHEMBL7531331 0.84 DHODH (0.55) CYP3A4PTGS1KMT2AMEN1ALDH1A1
SCHEMBL7539025 0.83 MEN1 (0.62) CYP3A4KMT2AMEN1ALDH1A1LMNA
SCHEMBL7568445 0.83 MEN1 (0.53) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
Sulfathiazole SCHEMBL7533713 0.83 LMNA (0.67) CYP3A4PTGS1SCN3ASCN5ASCN9A
Phthalylsulfathiazole SCHEMBL152662 0.82 CYP3A4 (1.00) CYP3A4PTGS1SCN3ASCN5ASCN9A
SCHEMBL7533705 0.81 SCN3A (0.56) CYP3A4PTGS1SCN3ASCN5ASCN9A
SCHEMBL7539041 0.80 MEN1 (0.53) KMT2AMEN1ALDH1A1MAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002028353-A2 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-11 WO claimed
WO-2002028353-A2 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-11 WO disclosed