SCHEMBL7533974

SCHEMBL7533974

CC(C)c1ccc(-n2nc(Cc3cccs3)c3c2CC(C)(C)CC3=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 11/20 0.47
HSP90AB1 P08238 4/20 0.42
SRC P12931 1/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
GAA P10253 1/20 0.37
HSP90AA1 P07900 2/20 0.37
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7534112 0.82 OPRM1 (0.50) OPRM1HSP90AB1SRCALDH1A1
SCHEMBL7479730 0.81 OPRM1 (0.54) OPRM1HSP90AB1SRCALDH1A1LMNA
SCHEMBL6770689 0.81 IDH1 (0.30) OPRM1LMNAKMT2A
SCHEMBL6772068 0.80 ALDH1A1 (0.57) OPRM1HSP90AB1ALDH1A1LMNANPSR1
SCHEMBL6766539 0.80 CCNA2 (0.35) SRCLMNAKMT2A
SCHEMBL6770401 0.76 OPRM1 (0.77) OPRM1HSP90AB1ALDH1A1LMNANPSR1
SCHEMBL6767006 0.76 OPRM1 (0.58) OPRM1HSP90AB1SRCHSP90AA1
SCHEMBL7533976 0.76 PARP1 (0.33) ALDH1A1LMNANPSR1KMT2A
SCHEMBL7537151 0.75 OPRM1 (0.54) OPRM1SRCALDH1A1LMNANPSR1
SCHEMBL6770500 0.73 OPRM1 (0.61) OPRM1HSP90AB1SRCHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed