SCHEMBL6767006

SCHEMBL6767006

CC(C)c1ccc(-n2nc(C(C)C)c3c2CC(C)(C)CC3=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 16/20 0.58
HSP90AB1 P08238 3/20 0.43
HSP90AA1 P07900 2/20 0.43
OPRD1 P41143 2/20 0.43
OPRK1 P41145 2/20 0.43
SRC P12931 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6769519 0.89 OPRM1 (0.54) OPRM1HSP90AB1HSP90AA1OPRD1OPRK1
SCHEMBL6168169 0.88 OPRM1 (0.53) OPRM1SRC
SCHEMBL6770401 0.87 OPRM1 (0.77) OPRM1HSP90AB1OPRD1OPRK1
SCHEMBL6770500 0.84 OPRM1 (0.61) OPRM1HSP90AB1HSP90AA1OPRD1OPRK1
SCHEMBL7479730 0.83 OPRM1 (0.54) OPRM1HSP90AB1HSP90AA1OPRD1OPRK1
SCHEMBL7537151 0.83 OPRM1 (0.54) OPRM1SRC
SCHEMBL6767149 0.83 OPRM1 (0.54) OPRM1HSP90AB1HSP90AA1OPRD1OPRK1
SCHEMBL6772068 0.82 ALDH1A1 (0.57) OPRM1HSP90AB1HSP90AA1OPRD1OPRK1
SCHEMBL7488247 0.81 OPRM1 (0.49) OPRM1HSP90AB1OPRD1OPRK1SRC
SCHEMBL7534112 0.79 OPRM1 (0.50) OPRM1HSP90AB1OPRD1OPRK1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed