SCHEMBL7536935

SCHEMBL7536935

CC(C)CCN(C(=O)NC1(C#N)CC1)C(=O)c1ccc(-c2csc(N3CCN(C(=O)O)CC3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSB P07858 13/20 0.49
CTSS P25774 13/20 0.49
CTSK P43235 5/20 0.49
KCNH2 Q12809 1/20 0.49
CTSL P07711 9/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MAPT P10636 5/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 4/20 0.40
MAPK1 P28482 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6182283 0.90 CTSB (0.44) CTSBCTSSCTSKKCNH2CTSL
SCHEMBL7616960 0.88 CTSS (0.45) CTSBCTSSCTSKKCNH2CTSL
SCHEMBL7544949 0.84 RAB9A (0.49) CTSBCTSSCTSKCTSLNPC1
SCHEMBL6182191 0.79 MAPT (0.55) CTSBCTSSCTSKCTSLNPC1
SCHEMBL6182260 0.79 CTSB (0.42) CTSBCTSSCTSKKCNH2CTSL
SCHEMBL6183519 0.78 ITGB3 (0.42)
SCHEMBL6183082 0.78 CTSS (0.46) CTSBCTSSCTSKCTSLNPC1
SCHEMBL7586301 0.75 MAPT (0.56) CTSBCTSSCTSKCTSLNPC1
SCHEMBL6183250 0.75 MAPT (0.44) CTSBCTSSCTSKCTSLNPC1
SCHEMBL7588285 0.74 MAPT (0.45) CTSBCTSSCTSKCTSLNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO disclosed