SCHEMBL7538007

SCHEMBL7538007

Cc1ccc(S(=O)(=O)N(C(=O)[C@H]2NC(C)(C)CS2)[C@@H](Cc2ccc(NC(=O)c3ccccc3)cc2)C(=O)O)cc1.Cc1ccc(S(=O)(=O)N(C(=O)[C@H]2NC(C)(C)CS2)[C@@H](Cc2ccc(O)cc2)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 2/20 0.46
MAPT P10636 9/20 0.44
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
LMNA P02545 5/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
MEN1 O00255 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA9 Q16790 2/20 0.36
CA2 P00918 1/20 0.36
THRB P10828 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGAV P06756 1/20 0.35
ITGA2B P08514 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6712491 0.97 MMP9 (0.48) MMP9MAPTITGB1ITGA4LMNA
SCHEMBL7189352 0.90 MMP9 (0.42) MMP9MAPTITGB1ITGA4LMNA
SCHEMBL6709350 0.89 ALDH1A1 (0.46) MMP9MAPTITGB1ITGA4SMN1; SMN2
SCHEMBL7421577 0.88 MMP9 (0.37) MMP9MAPTITGB1ITGA4LMNA
SCHEMBL6712429 0.88 LMNA (0.40) MMP9MAPTLMNASMN1; SMN2MEN1
SCHEMBL7320647 0.85 THRB (0.39) MMP9MAPTLMNASMN1; SMN2MEN1
SCHEMBL7319356 0.85 CA1 (0.37) MMP9MAPTLMNASMN1; SMN2MEN1
SCHEMBL5690666 0.83 MAPT (0.37) MMP9MAPTLMNASMN1; SMN2MEN1
SCHEMBL6714601 0.82 ALDH1A1 (0.45) MAPTSMN1; SMN2MEN1HTTKMT2A
SCHEMBL6708265 0.81 ALDH1A1 (0.44) MAPTSMN1; SMN2MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994896-A1 SULFONYLATED DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP disclosed
WO-1999006437-A1 SULFONYLATED DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS INC. (US) 1999-02-11 WO disclosed