SCHEMBL7538552

SCHEMBL7538552

COc1cccc(-n2nc(C(C)C)c3c2C(=O)CCC3C(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.42
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE4A P27815 4/20 0.38
PDE4B Q07343 4/20 0.38
PDE4C Q08493 4/20 0.38
PDE4D Q08499 4/20 0.38
ALOX5 P09917 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.36
HTT P42858 1/20 0.36
CYP3A4 P08684 1/20 0.36
GSK3B P49841 1/20 0.35
HSD11B1 P28845 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6771294 0.71 SRC (0.49) SRCRAB9ASMN1; SMN2L3MBTL1ALOX5
SCHEMBL6777339 0.71 CASP1 (0.39) SRCRAB9ASMN1; SMN2L3MBTL1KMT2A
SCHEMBL6775862 0.70 ABCG2 (0.39) SRCRAB9ASMN1; SMN2L3MBTL1KMT2A
SCHEMBL6777174 0.67 OPRM1 (0.58) SRC
SCHEMBL6770575 0.64 GPBAR1 (0.39) SRCRAB9ASMN1; SMN2L3MBTL1KMT2A
SCHEMBL6770505 0.64 OPRM1 (0.46) SRCRAB9ASMN1; SMN2L3MBTL1KMT2A
SCHEMBL6772956 0.62 SRC (0.49) SRCRAB9ASMN1; SMN2L3MBTL1ALOX5
SCHEMBL7480329 0.62 HRH2 (0.46) RAB9ASMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL6205595 0.62 HTT (0.46) RAB9ASMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL12988851 0.62 ADRB1 (0.58) RAB9ASMN1; SMN2KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed