SCHEMBL6770505

SCHEMBL6770505

COc1cccc(-n2nc(C)c3c2CC(C(C)C)CC3=O)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.46
MGLL Q99685 1/20 0.40
SRC P12931 1/20 0.40
DHODH Q02127 1/20 0.39
MAPT P10636 3/20 0.39
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38
CYP1A2 P05177 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6777339 0.89 CASP1 (0.39) OPRM1MGLLSRCDHODHMAPT
SCHEMBL6770575 0.88 GPBAR1 (0.39) OPRM1MGLLSRCDHODHMAPT
SCHEMBL6769819 0.87 OPRM1 (0.43) OPRM1SRCDHODHMAPTSMN1; SMN2
SCHEMBL6766674 0.87 RIPK2 (0.46) MGLLSRCDHODHMAPTRAB9A
SCHEMBL6772551 0.86 DHODH (0.37) MGLLSRCDHODHMAPTRAB9A
SCHEMBL6167296 0.86 HIF1A (0.47) OPRM1DHODHMAPTRAB9ASMN1; SMN2
SCHEMBL6766574 0.85 ALDH1A1 (0.39) MGLLDHODHMAPTRAB9ASMN1; SMN2
SCHEMBL6772063 0.85 OPRM1 (0.48) OPRM1MGLLSRCMAPTRAB9A
SCHEMBL6770636 0.81 RIPK2 (0.35) MGLLSRCDHODHMAPTRAB9A
SCHEMBL6770476 0.79 OPRM1 (0.45) OPRM1MGLLDHODHMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed