SCHEMBL7539838

SCHEMBL7539838

N#CC1Cc2cc(C(F)(F)F)ccc21

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.41
CHRNB2 P17787 3/20 0.40
CHRNA4 P43681 3/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
AADAT Q8N5Z0 1/20 0.36
SRD5A1 P18405 1/20 0.36
HTR2A P28223 5/20 0.36
HTR2C P28335 5/20 0.36
HTR2B P41595 5/20 0.36
HRH3 Q9Y5N1 2/20 0.35
NOTUM Q6P988 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583916 0.73 HSD17B10 (0.36) CHRNB2CHRNA4
SCHEMBL10850914 0.73 HTR2C (0.45) PNMTCHRNB2CHRNA4SRD5A1HTR2A
SCHEMBL3153525 0.73 TRPM5 (0.41) CHRNB2CHRNA4AADATSRD5A1
SCHEMBL2501307 0.73 CHRNB2 (0.42) CHRNB2CHRNA4HTR2A
SCHEMBL6984441 0.73 TRPV4 (0.33)
SCHEMBL3149299 0.72 DRD2 (0.41)
SCHEMBL5609696 0.70 SRD5A1 (0.49) PNMTCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL6986668 0.69
SCHEMBL16864134 0.69 SLC6A2 (0.38) SRD5A1HTR2AHTR2CHTR2B
SCHEMBL13976966 0.69 PNMT (0.41) PNMTCHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0940386-B1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2002-05-22 EP disclosed
US-6107345-A ANTIDEPRESSANT; PSYCHOLOGICAL DISORDERS ADIR ET COMPAGNIE (FR) 2000-08-22 US disclosed
EP-0940386-A1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-09-08 EP disclosed