SCHEMBL7540168

SCHEMBL7540168

BrCc1ccc2c(c1)Cc1cc(CBr)ccc1-2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
ALDH1A1 P00352 3/20 0.46
ATM Q13315 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
RAB9A P51151 5/20 0.41
NPC1 O15118 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP17A1 P05093 1/20 0.39
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
GPR84 Q9NQS5 1/20 0.36
HTT P42858 1/20 0.36
TRPA1 O75762 1/20 0.35
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29780668 0.90 TSHR (0.59) TSHRALDH1A1ATMNPSR1RAB9A
SCHEMBL7974044 0.90 TSHR (0.59) TSHRALDH1A1ATMNPSR1RAB9A
SCHEMBL6660057 0.86 AKR1B1 (0.39) TSHRALDH1A1ATMNPSR1ESR1
SCHEMBL8718934 0.84 ALDH1A1 (0.43) TSHRALDH1A1ATMNPSR1ESR1
SCHEMBL31468782 0.78 TRPA1 (0.36) TSHRALDH1A1ESR1ESR2MAPT
SCHEMBL11778412 0.77 ALDH1A1 (0.51) TSHRALDH1A1ATMNPSR1
SCHEMBL3284644 0.76 TSHR (0.42) TSHRALDH1A1MAPTHPGDCYP1A2
SCHEMBL29008215 0.76 CHEK1 (0.44) TSHRALDH1A1ATMNPSR1RAB9A
SCHEMBL4894905 0.76 ALDH1A1 (0.46) TSHRALDH1A1ATMNPSR1ESR1
SCHEMBL15625912 0.76 TSHR (0.63) TSHRALDH1A1ATMNPSR1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107245037-B Ladder-shaped macromolecule derivative and preparation method and application thereof 南京邮电大学 2020-02-07 CN disclosed
EP-1208088-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2002-05-29 EP disclosed
WO-2001010841-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2001-02-15 WO disclosed