SCHEMBL7536889

SCHEMBL7536889

FC(F)(F)C(F)(F)COc1cc2c(cc1C1=NCCN1)CCCC2

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 13/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8218198 0.79 NISCH (0.40) NISCHADRA2AADRA2BADRA2CKDM4E
SCHEMBL7543472 0.77 KDM4E (0.36) NISCHADRA2AADRA2BADRA2CKDM4E
Hydrochloric Acid SCHEMBL8218663 0.77 KDM4E (0.39) NISCHADRA2AADRA2BADRA2CKDM4E
Iodide SCHEMBL7537909 0.76 NOS3 (0.36) NISCHADRA2AADRA2BADRA2C
Iodide SCHEMBL7537243 0.73 ESR1 (0.36) NISCHADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL8207897 0.67 ADRA2A (0.47) NISCHADRA2AADRA2BADRA2C
SCHEMBL8196811 0.67 KDM4E (0.35) KDM4E
SCHEMBL8196356 0.66 HSD17B10 (0.42) KDM4E
SCHEMBL7534871 0.65 NISCH (0.64) NISCHADRA2AADRA2BADRA2CCYP1A2
SCHEMBL7538424 0.65 REN (0.33) NISCHADRA2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204644-A1 SYNTHESIS OF SUBSTITUTED AMIDINES ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2000078725-A1 SYNTHESIS OF SUBSTITUTED AMIDINES ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed
WO-2000078724-A2 IMIDAZOLINDERIVATIVES THEIR PREPARATION AND THEIR PHARMACEUTICAL USE ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed