SCHEMBL8208937

SCHEMBL8208937

COCCOc1c(C2=NCCN2)cc2c(c1Br)CCCC2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDCD1LG2 Q9BQ51 3/20 0.35
CD274 Q9NZQ7 3/20 0.35
NISCH Q9Y2I1 7/20 0.34
PARP1 P09874 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
MC4R P32245 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8218663 0.78 KDM4E (0.39) PDCD1LG2CD274NISCHKDM4E
SCHEMBL7543472 0.78 KDM4E (0.36) PDCD1LG2CD274NISCHKDM4E
SCHEMBL6820927 0.76 NISCH (0.59) PDCD1LG2CD274NISCHKDM4E
SCHEMBL8194455 0.71 ALDH1A1 (0.35) KDM4E
Hydrochloric Acid SCHEMBL8204086 0.71 CD274 (0.46) PDCD1LG2CD274NISCHMC4RKCNH2
SCHEMBL7538424 0.70 REN (0.33) PDCD1LG2CD274NISCHPARP1KDM4E
SCHEMBL8195029 0.70 MEN1 (0.43) PARP1
SCHEMBL6825218 0.70 KCNH2 (0.43) PDCD1LG2CD274NISCHMC4RKCNH2
SCHEMBL8198539 0.69 MC4R (0.49) PDCD1LG2CD274NISCHMC4RKCNH2
Hydrochloric Acid SCHEMBL7738758 0.69 KCNH2 (0.43) PDCD1LG2CD274NISCHMC4RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000078724-A2 IMIDAZOLINDERIVATIVES THEIR PREPARATION AND THEIR PHARMACEUTICAL USE ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed