SCHEMBL7545314

SCHEMBL7545314

C[C@@H](C(=O)N[C@H](C#N)CCc1ccccc1)N(C(=O)N1CCOCC1)c1ccc(F)cc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 17/20 0.62
CTSL P07711 2/20 0.53
CTSB P07858 1/20 0.53
CTSC P53634 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7546891 0.88 CTSS (0.60) CTSSCTSLCTSBCTSC
SCHEMBL7539922 0.84 CTSS (0.62) CTSSCTSLCTSBCTSC
SCHEMBL7393568 0.83 CTSS (0.60) CTSSCTSLCTSBCTSC
SCHEMBL7028324 0.78 CTSL (0.51) CTSSCTSLCTSBCTSC
SCHEMBL7378602 0.77 CTSS (0.45) CTSSCTSLCTSBCTSC
SCHEMBL6806938 0.75 CTSS (0.88) CTSSCTSLCTSB
SCHEMBL7062841 0.75 CTSS (1.00) CTSSCTSLCTSBCTSC
SCHEMBL8690335 0.74 CTSS (0.46) CTSSCTSLCTSBCTSC
SCHEMBL6800724 0.74 SMN1; SMN2 (0.46)
SCHEMBL6803089 0.74 CTSS (1.00) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed