SCHEMBL7546891

SCHEMBL7546891

C[C@@H](C(=O)N[C@H](C#N)CCc1ccccc1)N(C(=O)N1CCOCC1)c1ccc2ccccc2c1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSS P25774 17/20 0.60
CTSL P07711 2/20 0.51
CTSB P07858 1/20 0.51
CTSC P53634 2/20 0.45
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545314 0.88 CTSS (0.62) CTSSCTSLCTSBCTSC
SCHEMBL7393568 0.85 CTSS (0.60) CTSSCTSLCTSBCTSC
SCHEMBL7539922 0.83 CTSS (0.62) CTSSCTSLCTSBCTSCALDH1A1
SCHEMBL8696250 0.81 MMP2 (0.42) CTSSCTSLCTSBCTSCALDH1A1
SCHEMBL8696245 0.81 MMP2 (0.42) CTSSCTSLCTSBCTSCALDH1A1
SCHEMBL8696240 0.81 MMP2 (0.42) CTSSCTSLCTSBCTSCALDH1A1
SCHEMBL7358322 0.80 CTSL (0.62) CTSSCTSLCTSBCTSC
SCHEMBL7358323 0.80 CTSL (0.62) CTSSCTSLCTSBCTSC
SCHEMBL7358325 0.80 CTSL (0.62) CTSSCTSLCTSBCTSC
SCHEMBL7362208 0.80 CTSL (0.57) CTSSCTSLCTSBCTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed