SCHEMBL7547531

SCHEMBL7547531

Cc1ccccc1C(=S)c1ccnc(N)c1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.44
KDM5A P29375 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MYC P01106 2/20 0.39
PRKCI P41743 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
HPGD P15428 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9063741 0.88 NPC1 (0.39) NAPRTKDM5AKDM4CKDM5BNPC1
SCHEMBL7553608 0.86 NAPRT (0.46) NAPRTKDM5AKDM4CKDM5BMYC
SCHEMBL8798744 0.78 NAPRT (0.44) NAPRTKDM5AKDM4CKDM5BRAB9A
SCHEMBL8813141 0.78 NAPRT (0.44) NAPRTKDM5AKDM4CKDM5BNPC1
SCHEMBL7547894 0.76 MAPT (0.46) NAPRTKDM5AKDM4CKDM5BNOS3
Toluene SCHEMBL7547892 0.75 NAPRT (0.44) NAPRTKDM4CMYCPRKCIALDH1A1
SCHEMBL19857454 0.75 NAPRT (0.57) NAPRTKDM5AKDM4CKDM5BRAB9A
SCHEMBL20520335 0.74 NAPRT (0.47) NAPRTKDM4CRAB9APRKCINOS3
SCHEMBL8891362 0.73 ALDH1A1 (0.56) NAPRTMYCALDH1A1KDM4EPOLB
SCHEMBL1260539 0.73 NOS2 (0.52) NAPRTKDM5ANPC1RAB9ANOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed