SCHEMBL7547673

SCHEMBL7547673

NC(=O)c1cccnc1N1CCN(CCCN(c2ccncc2)c2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.46
DRD4 P21917 2/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2C P18825 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HRH1 P35367 1/20 0.43
DRD3 P35462 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
SLC6A4 P31645 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7546349 0.95 SIGMAR1 (0.48) SIGMAR1DRD4HTR1ADRD2ADRA2C
SCHEMBL7550443 0.81 SIGMAR1 (0.54) SIGMAR1DRD4HTR1ADRD2ADRA2C
Hydrochloric Acid SCHEMBL9602476 0.78 DRD3 (0.51) SIGMAR1DRD4HTR1ADRD2ADRA2C
Hydrochloric Acid SCHEMBL7541857 0.76 MAPT (0.61) SIGMAR1
Hydrochloric Acid SCHEMBL7549103 0.75 HTR1A (0.63) SIGMAR1DRD4HTR1ADRD2ADRA2C
Hydrochloric Acid SCHEMBL9601482 0.74 SIGMAR1 (0.48) SIGMAR1DRD4HTR1ADRD2ADRA2C
Hydrochloric Acid SCHEMBL9601471 0.74 SIGMAR1 (0.48) SIGMAR1DRD4HTR1ADRD2ADRA2C
SCHEMBL8878898 0.73 DRD2 (0.67) SIGMAR1DRD4HTR1ADRD2ADRA2C
Hydrochloric Acid SCHEMBL7544875 0.72 DRD2 (0.65) SIGMAR1DRD4HTR1ADRD2ADRA2C
SCHEMBL8037087 0.71 MAPK1 (0.58) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652867-B1 NOVEL PYRIDYL- AND PYRIMIDYLPIPERAZINE DERIVATIVES BIOVITRUM AB (SE) 2002-06-12 EP disclosed
US-6326371-B1 ANTISEROTININE AGENTS PHARMACIA AKTIEBOLAG (SE) 2001-12-04 US disclosed
US-5652240-A PSYCHOLOGICAL DISORDERS; ANXIOLYTIC AGENTS, ANTIDEPRESSANTS PHARMACIA AKTIEBOLAG (SE) 1997-07-29 US disclosed
EP-0652867-A1 NOVEL PYRIDYL- AND PYRIMIDYLPIPERAZINE DERIVATIVES Pharmacia & Upjohn Aktiebolag (SE) 1995-05-17 EP disclosed
WO-1994003430-A1 NOVEL PYRIDYL- AND PYRIMIDYLPIPERAZINE DERIVATIVES KABI PHARMACIA AB (SE) 1994-02-17 WO disclosed