SCHEMBL7550443

SCHEMBL7550443

Oc1cccnc1N1CCN(CCCN(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.54
HTR1A P08908 3/20 0.46
DRD2 P14416 3/20 0.46
HTR2A P28223 3/20 0.46
DRD3 P35462 3/20 0.46
DRD1 P21728 2/20 0.46
DRD5 P21918 1/20 0.46
HTR7 P34969 1/20 0.45
ADRA2C P18825 1/20 0.45
DRD4 P21917 1/20 0.45
HTR2C P28335 1/20 0.45
HRH1 P35367 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7546349 0.83 SIGMAR1 (0.48) SIGMAR1HTR1ADRD2HTR2ADRD3
Hydrochloric Acid SCHEMBL7549103 0.82 HTR1A (0.63) SIGMAR1HTR1ADRD2HTR2ADRD3
Hydrochloric Acid SCHEMBL7541857 0.81 MAPT (0.61) SIGMAR1
SCHEMBL7547673 0.81 SIGMAR1 (0.46) SIGMAR1HTR1ADRD2HTR2ADRD3
SCHEMBL8878898 0.80 DRD2 (0.67) SIGMAR1HTR1ADRD2HTR2ADRD3
SCHEMBL9601882 0.80 SIGMAR1 (0.56) SIGMAR1HTR1ADRD2HTR2ADRD3
Hydrochloric Acid SCHEMBL7544875 0.79 DRD2 (0.65) SIGMAR1HTR1ADRD2HTR2ADRD3
Hydrochloric Acid SCHEMBL11180176 0.74 SIGMAR1 (0.70) SIGMAR1HTR1ADRD2HTR2ADRD3
Hydrochloric Acid SCHEMBL11191151 0.73 SIGMAR1 (0.67) SIGMAR1
SCHEMBL11175427 0.73 SIGMAR1 (0.67) SIGMAR1HTR1ADRD2HTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652867-B1 NOVEL PYRIDYL- AND PYRIMIDYLPIPERAZINE DERIVATIVES BIOVITRUM AB (SE) 2002-06-12 EP disclosed
US-6326371-B1 ANTISEROTININE AGENTS PHARMACIA AKTIEBOLAG (SE) 2001-12-04 US disclosed
US-5652240-A PSYCHOLOGICAL DISORDERS; ANXIOLYTIC AGENTS, ANTIDEPRESSANTS PHARMACIA AKTIEBOLAG (SE) 1997-07-29 US disclosed
EP-0652867-A1 NOVEL PYRIDYL- AND PYRIMIDYLPIPERAZINE DERIVATIVES Pharmacia & Upjohn Aktiebolag (SE) 1995-05-17 EP disclosed
WO-1994003430-A1 NOVEL PYRIDYL- AND PYRIMIDYLPIPERAZINE DERIVATIVES KABI PHARMACIA AB (SE) 1994-02-17 WO disclosed