SCHEMBL7548608

SCHEMBL7548608

CCOC(=O)C#Cc1c(O)nc2ccccc2c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
ALDH1A1 P00352 2/20 0.45
POLB P06746 3/20 0.45
GLA P06280 1/20 0.45
TOP2A P11388 2/20 0.41
PRNP P04156 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
RXFP1 Q9HBX9 2/20 0.41
MAPT P10636 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 1/20 0.41
PDE10A Q9Y233 1/20 0.40
ABCB1 P08183 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545823 0.88 PDE10A (0.47) KDM4ESMN1; SMN2ALDH1A1POLBGLA
SCHEMBL7548798 0.80 SMN1; SMN2 (0.42) KDM4ESMN1; SMN2ALDH1A1POLBGLA
SCHEMBL7549915 0.75 PDE10A (0.41) KDM4ESMN1; SMN2ALDH1A1L3MBTL1CYP1A2
SCHEMBL26617516 0.74 SMN1; SMN2 (0.67) KDM4ESMN1; SMN2ALDH1A1POLBGLA
SCHEMBL7550340 0.74 PDE10A (0.41) KDM4EALDH1A1CYP1A2MEN1KMT2A
SCHEMBL7550385 0.71 KDM1A (0.39) KDM4EALDH1A1CYP1A2MAPTTDP1
SCHEMBL7915032 0.71 ALDH1A1 (0.56) KDM4EALDH1A1CYP1A2MAPTMEN1
SCHEMBL852513 0.71 GAA (0.50) SMN1; SMN2POLBTDP1MEN1KMT2A
SCHEMBL12267871 0.70 MAPT (0.43) KDM4EALDH1A1GLAL3MBTL1MAPT
SCHEMBL852937 0.70 ALDH1A1 (0.49) KDM4EALDH1A1POLBGLAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002046163-A2 QUINOLINE DERIVATIVES AND THEIR USE AS ANTI-EPILEPTICS WACKERNAGEL MICHAEL (DE) 2002-06-13 WO claimed
WO-2002046163-A2 QUINOLINE DERIVATIVES AND THEIR USE AS ANTI-EPILEPTICS WACKERNAGEL MICHAEL (DE) 2002-06-13 WO disclosed