SCHEMBL7548964

SCHEMBL7548964

NC(=O)c1cccnc1-c1c[nH]c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
ATM Q13315 1/20 0.56
HTR2C P28335 2/20 0.50
HTR2B P41595 2/20 0.50
HTR5A P47898 2/20 0.50
PIM1 P11309 2/20 0.49
PDE10A Q9Y233 1/20 0.46
CLK1 P49759 2/20 0.45
CDK5 Q00535 2/20 0.45
CDK5R1 Q15078 2/20 0.45
CAMKK2 Q96RR4 1/20 0.45
GSK3B P49841 2/20 0.45
DYRK1A Q13627 1/20 0.45
MAP3K14 Q99558 1/20 0.45
PDGFRB P09619 1/20 0.45
IMPDH2 P12268 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GPR84 Q9NQS5 1/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7053843 0.84 CAMKK2 (0.63) PIM1CDK5CDK5R1CAMKK2GSK3B
SCHEMBL29822183 0.82 NUDT1 (0.50) ALDH1A1ATMPIM1CDK5GSK3B
SCHEMBL28305303 0.79 ALDH1A1 (0.67) ALDH1A1ATMPIM1MAPK1GPR84
SCHEMBL3673827 0.79 ALDH1A1 (0.67) ALDH1A1ATMPIM1MAPK1GPR84
SCHEMBL18982934 0.76 PIM1 (0.53) ALDH1A1ATMHTR2CHTR2BHTR5A
SCHEMBL31032166 0.75 PARP1 (0.55) ALDH1A1MAPK1HSD17B10MEN1KMT2A
SCHEMBL28677807 0.75 PARP1 (0.55) ALDH1A1MAPK1HSD17B10MEN1KMT2A
SCHEMBL30108279 0.75 PARP1 (0.55) ALDH1A1MAPK1HSD17B10MEN1KMT2A
SCHEMBL7382969 0.75 ALDH1A1 (0.56) ALDH1A1ATMPIM1GSK3BDYRK1A
SCHEMBL28035470 0.75 CSNK1A1 (0.49) ALDH1A1HSD17B10MEN1KMT2ACSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785789-B1 DIAZEPINO-INDOLES AS PHOSPHODIESTERASE IV INHIBITORS PFIZER (FR) 2002-09-11 EP disclosed