SCHEMBL7053843

SCHEMBL7053843

NC(=O)c1cccnc1-c1c[nH]c2ncccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 3/20 0.63
NUDT1 P36639 1/20 0.52
MAP2K1 Q02750 1/20 0.50
RPS6KA5 O75582 1/20 0.49
NEK2 P51955 1/20 0.48
PLK1 P53350 1/20 0.48
CDK2 P24941 4/20 0.48
CDC7 O00311 3/20 0.48
TGFBR1 P36897 2/20 0.48
PDPK1 O15530 2/20 0.48
CCNT1 O60563 1/20 0.48
CCNA2 P20248 1/20 0.48
CDK9 P50750 1/20 0.48
CCNA1 P78396 1/20 0.48
CDK5 Q00535 1/20 0.48
CDK5R1 Q15078 1/20 0.48
IKBKE Q14164 1/20 0.47
TBK1 Q9UHD2 1/20 0.46
CCNE1 P24864 2/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30563455 0.86 NUDT1 (0.67) CAMKK2NUDT1MAP2K1NEK2PLK1
SCHEMBL7548964 0.84 ALDH1A1 (0.56) CAMKK2PDPK1CDK5CDK5R1PIM1
SCHEMBL586850 0.82 MAP2K1 (0.67) CAMKK2NUDT1MAP2K1NEK2CDK2
Water SCHEMBL15530974 0.80 MAP2K1 (0.65) CAMKK2NUDT1MAP2K1NEK2PLK1
Hydrochloric Acid SCHEMBL5263201 0.80 MAP2K1 (0.65) CAMKK2NUDT1MAP2K1NEK2CDK2
SCHEMBL1820660 0.78 ADORA2A (0.61) CAMKK2NUDT1MAP2K1NEK2PLK1
SCHEMBL4374583 0.77 CAMKK2 (0.62) CAMKK2RPS6KA5NEK2PLK1CDK2
SCHEMBL8939859 0.77 CAMKK2 (1.00) CAMKK2MAP2K1RPS6KA5NEK2PLK1
SCHEMBL30320851 0.76 CAMKK2 (0.55) CAMKK2MAP2K1RPS6KA5CDK2CDC7
SCHEMBL5618155 0.76 TGFBR1 (0.71) CAMKK2MAP2K1RPS6KA5CDK2CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028724-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO claimed
WO-2003028724-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed