SCHEMBL7549906

SCHEMBL7549906

[N-]=[N+]=C1C(=O)Oc2cc(O)ccc2C1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 4/20 0.51
MAOA P21397 4/20 0.51
MAOB P27338 4/20 0.51
CISD1 Q9NZ45 2/20 0.50
MEN1 O00255 7/20 0.47
KMT2A Q03164 7/20 0.47
USP2 O75604 2/20 0.47
CASP3 P42574 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
RECQL P46063 3/20 0.47
POLB P06746 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 2/20 0.47
GAA P10253 2/20 0.47
MAPT P10636 2/20 0.47
PSMD14 O00487 1/20 0.47
AURKA O14965 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545914 0.87 TYR (0.49) TYRMAOAMAOBCISD1MEN1
SCHEMBL6984812 0.81 MAOA (0.57) TYRMAOAMAOBCISD1MEN1
SCHEMBL6670897 0.78 STK17B (0.47) TYRMAOAMAOBCISD1MEN1
SCHEMBL7552791 0.74 MAOB (0.54) MAOAMAOBRAB9ANPC1
SCHEMBL7567696 0.72 STK17B (0.42) TYRMAOAMAOBCISD1MEN1
SCHEMBL23728337 0.70 MAOA (0.54) TYRMAOAMAOBCISD1MEN1
SCHEMBL14259795 0.70 MAOA (0.49) TYRMAOAMAOBCISD1MEN1
SCHEMBL2114477 0.70 MAOA (0.49) TYRMAOAMAOBCISD1MEN1
SCHEMBL7578571 0.70 STK17B (0.39) TYRMAOAMAOBMEN1KMT2A
SCHEMBL7547313 0.69 TYR (0.47) TYRMAOAMAOBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968202-B1 Process for preparing photoactive coumarin dervatives CLARIANT FINANCE BVI LTD (VG) 2002-07-03 EP disclosed
EP-0968202-B1 Process for preparing photoactive coumarin dervatives CLARIANT FINANCE BVI LTD (VG) 2002-07-03 EP disclosed
EP-0977747-B1 PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT FINANCE BVI LTD (VG) 2002-06-12 EP disclosed
EP-0977747-B1 PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT FINANCE BVI LTD (VG) 2002-06-12 EP disclosed
CN-1254338-A Process for preparing photoactive coumarin derivatives HOECHST CELANESE CORP (CH) 2000-05-24 CN disclosed
CN-1251584-A Photoactive coumarin derivatives HOECHST CELANESE INTERNATIONAL (CH) 2000-04-26 CN disclosed
EP-0977747-A1 PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 2000-02-09 EP disclosed
EP-0977747-A1 PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 2000-02-09 EP disclosed
EP-0968202-A1 PROCESS FOR PREPARING PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 2000-01-05 EP disclosed
EP-0968202-A1 PROCESS FOR PREPARING PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 2000-01-05 EP disclosed
WO-1998039317-A1 PROCESS FOR PREPARING PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 1998-09-11 WO disclosed
WO-1998039317-A1 PROCESS FOR PREPARING PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 1998-09-11 WO disclosed
WO-1998039319-A1 PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 1998-09-11 WO disclosed
WO-1998039319-A1 PHOTOACTIVE COUMARIN DERIVATIVES CLARIANT INTERNATIONAL LTD. (CH) 1998-09-11 WO disclosed
US-5726296-A PHOTORESISTS HOECHST CELANESE CORP. (US) 1998-03-10 US disclosed
US-5726296-A PHOTORESISTS HOECHST CELANESE CORP. (US) 1998-03-10 US disclosed
US-5726295-A Photoactive coumarin derivatives HOECHST CELANESE CORP. (US) 1998-03-10 US disclosed
US-5726295-A Photoactive coumarin derivatives HOECHST CELANESE CORP. (US) 1998-03-10 US disclosed