SCHEMBL7557478

SCHEMBL7557478

Nc1cc(S(=O)(=O)Nc2ccccc2NC(=O)Nc2ccccc2Br)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 7/20 0.53
CXCR1 P25024 6/20 0.53
MAPT P10636 4/20 0.52
NPSR1 Q6W5P4 1/20 0.52
PTGES2 Q9H7Z7 2/20 0.48
MEN1 O00255 5/20 0.47
LMNA P02545 5/20 0.47
KMT2A Q03164 5/20 0.47
PKM P14618 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
IDH1 O75874 1/20 0.46
HTT P42858 2/20 0.45
MAPK1 P28482 1/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GRIK1 P39086 1/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7494404 0.82 POLB (0.51) CXCR2CXCR1MAPTPTGES2MEN1
SCHEMBL5737217 0.78 GAA (0.66) MAPTNPSR1PTGES2MEN1LMNA
SCHEMBL10695037 0.77 MEN1 (0.73) MEN1LMNAKMT2AGAAKDM4E
SCHEMBL5594928 0.76 DDX3X (0.63) CXCR2CXCR1MAPTMEN1LMNA
SCHEMBL7951681 0.75 PTGES2 (0.59) CXCR2CXCR1MAPTPTGES2MEN1
SCHEMBL5595046 0.75 HTT (0.60) MEN1LMNAKMT2AHTTGAA
SCHEMBL5595427 0.75 CA12 (0.52) PTGES2MEN1LMNAKMT2ACA12
SCHEMBL15145842 0.74 MEN1 (0.64) MAPTMEN1LMNAKMT2ACA2
SCHEMBL13577027 0.74 LMNA (0.62) MAPTMEN1LMNAKMT2APKM
SCHEMBL5595863 0.74 MEN1 (0.49) CXCR2CXCR1MAPTNPSR1PTGES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020128321-A1 IL-8 receptor antagonists SMITHKLINE BEECHAM CORPORATION 2002-09-12 US disclosed
US-6262113-B1 HYDROXY- OR MERCAPTO-PHENYLUREAS SMITHKLINE BEECHAM CORPORATION 2001-07-17 US disclosed
US-6211373-B1 Phenyl urea antagonists of the IL-8 receptor SMITHKLINE BEECHAM CORPORATION 2001-04-03 US disclosed
US-5780483-A IL-8 receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 1998-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020128321-A1 IL-8 receptor antagonists CXCL8, CCR8, IL1RN CXCR2 15/4885CXCR1 21/4885MAPT 698/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.