SCHEMBL7562355

SCHEMBL7562355

Cc1cccc2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)NC(C(=O)CC(=O)c3c(Cl)cccc3Cl)C(=O)C(=O)O)c(CC(C)C)c12

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 3/20 0.39
ITGB2 P05107 3/20 0.38
ICAM1 P05362 3/20 0.38
ITGAL P20701 3/20 0.38
PYGL P06737 1/20 0.34
ITGB1 P05556 5/20 0.33
ITGA4 P13612 5/20 0.33
ITGB7 P26010 2/20 0.33
ITGA2 P17301 1/20 0.33
CAPN1 P07384 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7564924 0.80 KDM4E (0.36) ITGB2ICAM1ITGAL
SCHEMBL7536650 0.76 MMP2 (0.38) ITGB2ICAM1ITGALCAPN1
SCHEMBL7201321 0.76 PSMB5 (0.40) PSMB5ITGB2ICAM1ITGALPYGL
SCHEMBL7536449 0.72 MMP2 (0.36)
SCHEMBL7543444 0.70 CASP3 (0.49)
SCHEMBL7432924 0.68 FBP1 (0.50)
SCHEMBL7535627 0.66 CASP3 (0.40)
SCHEMBL17969599 0.65 FEN1 (0.42) ITGB2ICAM1ITGAL
SCHEMBL20815821 0.62 PSMB5 (0.55) PSMB5ITGB2ICAM1ITGALITGB1
SCHEMBL20815818 0.62 PSMB5 (0.55) PSMB5ITGB2ICAM1ITGALITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159291-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-12-05 EP disclosed
WO-2001000658-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2001-01-04 WO disclosed