SCHEMBL7536650

SCHEMBL7536650

Cc1cccc2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)NC(CC(=O)O)C(=O)CBr)c(CC(C)C)c12

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP1 P03956 1/20 0.38
EDNRA P25101 1/20 0.37
CTNNB1 P35222 1/20 0.37
ANPEP P15144 2/20 0.35
ERAP2 Q6P179 1/20 0.34
CNR2 P34972 1/20 0.34
CTSL P07711 2/20 0.34
CLPP Q16740 2/20 0.34
CCKBR P32239 3/20 0.34
GAA P10253 1/20 0.33
CAPN1 P07384 1/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33
ITGAL P20701 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7535627 0.90 CASP3 (0.40) MMP2MMP9MMP8
SCHEMBL7536449 0.86 MMP2 (0.36) MMP2MMP9MMP8MMP1EDNRA
SCHEMBL7543444 0.84 CASP3 (0.49)
SCHEMBL8606968 0.81 CASP3 (0.41)
SCHEMBL7562355 0.76 PSMB5 (0.39) CAPN1ITGB2ICAM1ITGAL
SCHEMBL7538962 0.76 CASP3 (0.58)
SCHEMBL7535127 0.75 CASP3 (0.47)
SCHEMBL7540320 0.74 CASP3 (0.49)
SCHEMBL27563383 0.72 CTSL (0.37) MMP2MMP9MMP8MMP1EDNRA
SCHEMBL7200894 0.72 CTSL (0.37) MMP2MMP9MMP8MMP1EDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159291-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-12-05 EP disclosed
WO-2001000658-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2001-01-04 WO disclosed