SCHEMBL7562480

SCHEMBL7562480

O=C(Cn1ccnc1)N[CH]c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
HMOX2 P30519 1/20 0.51
KDM4E B2RXH2 1/20 0.50
AHR P35869 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TBXAS1 P24557 2/20 0.48
CYP19A1 P11511 4/20 0.48
CYP11B1 P15538 2/20 0.47
CYP11B2 P19099 2/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
MAPT P10636 1/20 0.47
QPCT Q16769 1/20 0.47
CYP4Z1 Q86W10 1/20 0.47
QPCTL Q9NXS2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10247217 0.78 SMN1; SMN2 (0.62) ALDH1A1HMOX2TBXAS1CYP19A1CYP11B1
SCHEMBL21076446 0.78 MGLL (0.62) ALDH1A1HMOX2KDM4EAHRNPSR1
Hydrochloric Acid SCHEMBL411425 0.77 SMN1; SMN2 (0.61) ALDH1A1HMOX2TBXAS1CYP19A1CYP11B1
Biphenyl SCHEMBL27824074 0.75 ALDH1A1 (0.76) ALDH1A1HMOX2CYP19A1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL11635603 0.74 TBXAS1 (0.58) ALDH1A1HMOX2TBXAS1CYP1A2CYP3A4
SCHEMBL11238973 0.73 HMOX2 (0.64) ALDH1A1HMOX2TBXAS1CYP19A1CYP11B1
SCHEMBL20830350 0.72 HMOX2 (0.49) ALDH1A1HMOX2TBXAS1CYP19A1CYP11B1
SCHEMBL1509735 0.72 CYP19A1 (0.71) ALDH1A1TBXAS1CYP19A1CYP11B1CYP11B2
SCHEMBL77978 0.72
SCHEMBL11131296 0.71 CYP19A1 (0.70) TBXAS1CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002067654-A3 6-SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-10-31 WO claimed
EP-1121363-A2 6-SUBSTITUTED PYRAZOLO 3,4-d]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS Du Pont Pharmaceuticals Company (US) 2001-08-08 EP claimed
WO-2000021926-A2 6-SUBSTITUTED PYRAZOLO[3,4-d]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 2000-04-20 WO claimed
WO-2002067654-A3 6-SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-10-31 WO disclosed