SCHEMBL756393

SCHEMBL756393

O=C(O)N1CCOc2ccc(Oc3cccc(-c4cncs4)c3)cc2S1(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR142 Q7Z601 5/20 0.38
MGLL Q99685 1/20 0.37
PLAUR Q03405 1/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
FAAH O00519 2/20 0.33
GAA P10253 2/20 0.32
WNT1 P04628 3/20 0.32
GSK3B P49841 3/20 0.32
DYRK1A Q13627 3/20 0.32
PIK3CD O00329 1/20 0.32
NAAA Q02083 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL760502 0.82 FFAR1 (0.38) GPR142FAAHGAAPIK3CDHCRTR1
SCHEMBL759900 0.81 FAAH (0.44) GPR142FAAHNAAA
SCHEMBL765578 0.79 KEAP1 (0.42) GPR142MGLLDYRK1APIK3CDHCRTR1
SCHEMBL759673 0.74 MAPT (0.43) FAAH
SCHEMBL782217 0.73 GPR119 (0.38) GPR142GAAPIK3CDHCRTR1HCRTR2
SCHEMBL765579 0.73 LMNA (0.51) GPR142GAA
SCHEMBL758615 0.71 TDP1 (0.45) FAAH
SCHEMBL781918 0.71 FAAH (0.39) GPR142FAAHNAAA
SCHEMBL782067 0.70 BACE1 (0.38) GPR142MGLLFAAH
SCHEMBL760249 0.67 LMNA (0.37) PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431360-B1 Derivatives of dihydrobenzoxathiazepine, method of preparing same and pharmaceutical compositions containing them as well as their uses as modulators of AMPA receptors SERVIER LAB (FR) 2013-04-17 EP disclosed
EP-2431360-A1 Derivatives of dihydrobenzoxathiazepine, method of preparing same and pharmaceutical compositions containing them as well as their uses as modulators of AMPA receptors Les Laboratoires Servier (FR) 2012-03-21 EP disclosed