SCHEMBL7564002

SCHEMBL7564002

COc1ccc(N(C)C(=O)c2c(O)c3c(N(C)C)c(C)ccc3[nH]c2=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
GPBAR1 Q8TDU6 2/20 0.38
PADI4 Q9UM07 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HDAC4 P56524 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX12 P18054 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RECQL P46063 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828560 0.79 GPBAR1 (0.40) HSP90AA1PDK1PDK2PDK3PDK4
SCHEMBL9187433 0.79 ALDH1A1 (0.47) HSP90AA1PDK1PDK2PDK3PDK4
SCHEMBL9186522 0.79 KDM4E (0.51) PADI4LMNAMAPTALDH1A1KDM4E
SCHEMBL6204567 0.76 HDAC4 (0.49) GPBAR1MAPTALDH1A1HDAC4
SCHEMBL7557817 0.76 GPBAR1 (0.40) GPBAR1CYP3A4CYP2C19
SCHEMBL7558468 0.76 GPBAR1 (0.38) GPBAR1MAPTKDM4E
SCHEMBL6202118 0.75 MEN1 (0.43) ALDH1A1KDM4ECYP2C9
SCHEMBL7829858 0.74 MAPT (0.48) PDK2TP53MAPTALDH1A1KDM4E
SCHEMBL11983220 0.74 HDAC4 (0.51) GPBAR1MAPTALDH1A1KDM4EHDAC4
SCHEMBL7818937 0.73 PTGS2 (0.44) GPBAR1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224172-A1 DRUGS FOR THE TREATMENT OF MALIGNANT TUMOURS Active Biotech AB (SE) 2002-07-24 EP claimed
WO-2001030758-A1 DRUGS FOR THE TREATMENT OF MALIGNANT TUMOURS ACTIVE BIOTECH AB (SE) 2001-05-03 WO claimed