SCHEMBL756450

SCHEMBL756450

COC(=O)ON1C(=O)CCC1=O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
BRD4 O60885 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
HTT P42858 1/20 0.32
GAA P10253 1/20 0.32
GLA P06280 1/20 0.32
CYP1A2 P05177 1/20 0.32
HIF1A Q16665 1/20 0.32
POLB P06746 1/20 0.31
THRB P10828 1/20 0.31
PARL Q9H300 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15371562 0.86 KMT2A (0.32) MGLLKMT2AATMGAA
SCHEMBL19447705 0.86 KMT2A (0.32) MGLLKMT2AATM
SCHEMBL17447 0.85 MGLL (0.37) MGLLGLAPARL
SCHEMBL9546740 0.82 MGLL (0.33) MGLLKMT2AATMALDH1A1HPGD
SCHEMBL9546488 0.82 MGLL (0.33) MGLLKMT2AATMALDH1A1HPGD
SCHEMBL2139612 0.81 MGLL (0.35) MGLLPARL
SCHEMBL15591345 0.81 CCNE1 (0.34) MGLLBRD4
SCHEMBL18947917 0.81 MGLL (0.31) MGLL
SCHEMBL726706 0.81 MGLL (0.37) MGLLKMT2AATMALDH1A1HPGD
SCHEMBL21582363 0.79 BRD4 (0.35) KMT2AATMBRD4ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 340 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114890916-A Preparation method of N-methoxycarbonyl-L-tert-leucine 常州吉恩药业有限公司 2022-08-12 CN claimed
CN-114685316-A MOC-L-valine synthesis process 常州吉恩药业有限公司 2022-07-01 CN claimed
EP-4649086-A1 PROTEASE INHIBITORS FOR TREATING OR PREVENTING CORONAVIRUS INFECTION Merck Sharp & Dohme LLC (US) 2025-11-19 EP disclosed
EP-4622959-A1 2-AMINO-N-(4-AMINO-3,4-DIOXO-1-(2-OXOPYRROLIDIN-3-YL)BUTAN-2-YL)BENZAMIDE DERIVATIVES AS PROTEASE INHIBITORS FOR TREATING OR PREVENTING CORONAVIRUS INFECTION Merck Sharp & Dohme LLC (US) 2025-10-01 EP disclosed
EP-3706747-B1 PRMT5 INHIBITORS MERCK SHARP & DOHME LLC (US) 2025-09-03 EP disclosed
WO-2025094035-A1 TOLL-LIKE RECEPTOR AGONISTS AND CONJUGATES THEREOF PFIZER INC. (US) 2025-05-08 WO disclosed
US-20240269293-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF OD THERAPEUTICS LIMITED (CN) 2024-08-15 US disclosed
WO-2024151465-A1 PROTEASE INHIBITORS FOR TREATING OR PREVENTING CORONAVIRUS INFECTION MERCK SHARP & DOHME LLC (US) 2024-07-18 WO disclosed
US-20240228535-A1 PROTEASE INHIBITORS FOR TREATING OR PREVENTING CORONAVIRUS INFECTION MERCK SHARP & DOHME LLC (US) 2024-07-11 US disclosed
US-20240228535-A1 PROTEASE INHIBITORS FOR TREATING OR PREVENTING CORONAVIRUS INFECTION MERCK SHARP & DOHME LLC (US) 2024-07-11 US disclosed
WO-2024112621-A1 2-AMINO-N-(4-AMINO-3,4-DIOXO-1-(2-OXOPYRROLIDIN-3-YL)BUTAN-2-YL)BENZAMIDE DERIVATIVES AS PROTEASE INHIBITORS FOR TREATING OR PREVENTING CORONAVIRUS INFECTION MERCK SHARP & DOHME LLC (US) 2024-05-30 WO disclosed
WO-2006012725-A1 LYSINE BASED COMPOUNDS AMBRILIA BIOPHARMA INC. (CA) 2006-02-09 WO disclosed
US-20060025592-A1 Lysine based compounds TAIMED BIOLOGICS, INC. (TW) 2006-02-02 US disclosed
CN-1690193-A Use of methioninase in anti-methionine and anti-homocysteine chemotherapy ANTICANCER INC (US) 2005-11-02 CN disclosed
EP-1575914-A1 AROMATIC DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS Procyon Biopharma Inc. (CA) 2005-09-21 EP disclosed
CN-1589257-A N-methyl-homocysteine and application and preparation method thereof SCHERING AG (DE) 2005-03-02 CN disclosed
WO-2004056764-A1 AROMATIC DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS PROCYON BIOPHARMA INC. (CA) 2004-07-08 WO disclosed
US-6632816-B1 Aromatic derivatives as HIV aspartyl protease inhibitors PHARMACOR INC. (CA) 2003-10-14 US disclosed
WO-1994018229-A1 1,2,4-TRIAZINONE DERIVATIVES AND THEIR USE IN THERAPY FISONS CORPORATION (US) 1994-08-18 WO disclosed
CN-1053607-A The human immunity that is used for the treatment of AIDS lacks the inhibitor of virus protease MERCK & CO INC (US) 1991-08-07 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240269293-A1 PROTEIN-MACROMOLECULE CONJUGATES AND METHODS OF USE THEREOF CD44, MACROD1, MSN MGLL 2707/4885KMT2A 2714/4885ATM 668/4885
US-20240228535-A1 PROTEASE INHIBITORS FOR TREATING OR PREVENTING CORONAVIRUS INFECTION PRSS1, PRSS2, ACE2 MGLL 1422/4885KMT2A 3149/4885ATM 2521/4885
US-20060025592-A1 Lysine based compounds DOT1L, H1-2, H1-0 MGLL 1640/4885KMT2A 12/4885ATM 1593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.