SCHEMBL7564626

SCHEMBL7564626

NC(=O)c1ccccc1C(=O)NCCc1ccc2ccccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.50
LMNA P02545 2/20 0.50
CES2 O00748 1/20 0.48
NPC1 O15118 4/20 0.47
RAB9A P51151 2/20 0.47
PKM P14618 2/20 0.46
NAMPT P43490 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
CYP1A2 P05177 1/20 0.46
ALDH1A1 P00352 2/20 0.45
HTT P42858 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3235358 0.84 ESRRG (0.61) MAPTCES2NPC1RAB9APKM
SCHEMBL23832296 0.83 HPGD (0.58) CES2NPC1RAB9AALDH1A1MEN1
SCHEMBL6198665 0.82 CES2 (0.54) MAPTLMNACES2PKMNAMPT
SCHEMBL27592472 0.82 NPC1 (0.67) MAPTLMNANPC1RAB9AALDH1A1
SCHEMBL3235573 0.80 PKM (0.58) MAPTCES2NPC1RAB9APKM
SCHEMBL5969148 0.80 ESRRG (0.60) NPC1RAB9ACYP1A2MEN1KMT2A
SCHEMBL6903284 0.78 TSHR (0.58) MAPTLMNANPC1RAB9AALDH1A1
SCHEMBL3232164 0.78 ESRRG (0.59) MAPTCES2NPC1RAB9ARXFP1
SCHEMBL2732841 0.77 CYP1A2 (0.58) MAPTLMNACES2PKMRXFP1
SCHEMBL761158 0.76 KDM4E (0.61) MAPTLMNACES2PKMRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002020437-A2 BASIC COMPOUNDS CONTAINING TERTIARY AMIDES WITH ACTIVITY ON TACHYKININ RECEPTORS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MENARINI RICERCHE S.P.A. (IT) 2002-03-14 WO claimed
WO-2002020437-A2 BASIC COMPOUNDS CONTAINING TERTIARY AMIDES WITH ACTIVITY ON TACHYKININ RECEPTORS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MENARINI RICERCHE S.P.A. (IT) 2002-03-14 WO disclosed