SCHEMBL7564705

SCHEMBL7564705

CCOC(=O)C(NC(=O)OC(C)(C)C)C1CCc2ccccc2NC1=O

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.46
CALCRL Q16602 1/20 0.41
EPHX2 P34913 1/20 0.40
SCN9A Q15858 5/20 0.39
CCKAR P32238 1/20 0.39
CCKBR P32239 1/20 0.39
CTSL P07711 2/20 0.38
SMYD3 Q9H7B4 1/20 0.38
CTSK P43235 2/20 0.37
CTSB P07858 1/20 0.37
DRD2 P14416 2/20 0.37
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31758027 0.83 DRD2 (0.41) IDO1SCN9ACTSLCTSKCTSB
SCHEMBL31757665 0.83 DRD2 (0.41) IDO1SCN9ACTSLCTSKCTSB
SCHEMBL7571221 0.83 IDO1 (0.46) IDO1EPHX2CCKARCCKBRCTSL
SCHEMBL7565993 0.82 IDO1 (0.52) IDO1CALCRLEPHX2CCKARCCKBR
SCHEMBL7567176 0.81 EPHX2 (0.53) IDO1EPHX2SCN9ACTSLSMYD3
SCHEMBL11118986 0.79 IDO1 (0.46) IDO1SCN9ACCKARCCKBRCTSL
SCHEMBL7543362 0.78 ALDH1A1 (0.43) ALDH1A1MAPTL3MBTL1
SCHEMBL11118093 0.78 ALDH1A1 (0.43) ALDH1A1MAPTL3MBTL1
SCHEMBL15414265 0.77 SCN9A (0.47) IDO1EPHX2SCN9A
SCHEMBL15414268 0.77 SCN9A (0.47) IDO1EPHX2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0072352-A1 Benzazepin-2-ones, process for their preparation, pharmaceutical preparations containing these compounds and the compounds for therapeutical use CIBA-GEIGY AG (CH) 1983-02-16 EP disclosed