SCHEMBL7565671

SCHEMBL7565671

COc1cc(OC)cc(C(=O)NCC(C(=O)NCC#N)C2CCCCC2)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.52
ALDH1A1 P00352 3/20 0.50
POLB P06746 1/20 0.50
LMNA P02545 1/20 0.47
CTSL P07711 3/20 0.47
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.45
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
NPC1 O15118 2/20 0.42
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
RAB9A P51151 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5527570 0.90 CTSL (0.53) ALDH1A1LMNACTSLHPGDGAA
SCHEMBL5529207 0.89 ALDH1A1 (0.54) KMT2AMEN1ALDH1A1LMNACTSL
SCHEMBL5530631 0.88 TDP1 (0.56) KMT2AMEN1ALDH1A1POLBCTSL
SCHEMBL5525342 0.84 CTSL (0.60) ALDH1A1LMNACTSLGAACTSB
SCHEMBL5528969 0.83 PKM (0.56) KMT2AMEN1ALDH1A1LMNACTSL
SCHEMBL5522184 0.82 CTSL (0.56) POLBLMNACTSLHPGDCTSB
SCHEMBL5521620 0.82 CTSL (0.56) CTSLCTSBCTSSCTSKNPC1
SCHEMBL5525451 0.82 CTSL (0.49) CTSLCTSBCTSSCTSKNPC1
SCHEMBL5529016 0.81 RAB9A (0.59) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL6690368 0.81 CTSS (0.58) KMT2AMEN1ALDH1A1POLBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178958-A2 N-CYANOMETHYL AMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-02-13 EP disclosed
WO-2000055125-A2 N-CYANOMETHYL AMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed