SCHEMBL7572580

SCHEMBL7572580

COC(=O)C(N)(CC#Cc1ccccc1)S(=O)(=O)c1ccc(I)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 14/20 0.39
MMP2 P08253 11/20 0.39
MMP3 P08254 11/20 0.39
MMP1 P03956 4/20 0.39
MMP9 P14780 2/20 0.39
MMP8 P22894 1/20 0.39
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
CA7 P43166 1/20 0.38
HTT P42858 1/20 0.37
F2 P00734 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7502964 0.88 MMP13 (0.50) MMP13MMP2MMP3MMP1MMP9
SCHEMBL7502278 0.86 MMP13 (0.55) MMP13MMP2MMP3MMP1MMP9
SCHEMBL7587417 0.86 ALDH1A1 (0.41) CA12CA1CA2CA9HTT
SCHEMBL7502706 0.86 MMP13 (0.50) MMP13MMP2MMP3MMP1MMP9
SCHEMBL7451550 0.82 MMP2 (0.46) MMP13MMP2MMP3MMP1CA12
SCHEMBL7450581 0.81 MMP2 (0.49) MMP13MMP2MMP3MMP1MMP9
SCHEMBL7898486 0.79 MMP2 (0.56) MMP13MMP2MMP3MMP1MMP9
SCHEMBL7512865 0.78 KMT2A (0.39) MMP13MMP2MMP3MMP1MMP9
SCHEMBL7547380 0.77 MMP2 (0.41) MMP13MMP2MMP3MMP1HTT
SCHEMBL7516820 0.76 MMP13 (0.54) MMP13MMP2MMP3MMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165501-A1 ALKENYL- AND ALKYNYL-CONTAINING METALLOPROTEASE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2002-01-02 EP disclosed
US-6197770-B1 ENZYME INHIBITORS; ANTIARTHRITIC AGENTS; BONE DISORDERS THE PROCTER & GAMBLE CO. 2001-03-06 US disclosed
WO-2000051975-A1 ALKENYL- AND ALKYNYL-CONTAINING METALLOPROTEASE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2000-09-08 WO disclosed