SCHEMBL7572810

SCHEMBL7572810

CC(C)=CCOc1cc(N=C=S)ccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
KDM4E B2RXH2 3/20 0.34
MTNR1A P48039 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
TRPA1 O75762 1/20 0.34
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
PTGES O14684 2/20 0.34
P2RY6 Q15077 2/20 0.33
RAD1 O60671 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13861946 0.76 L3MBTL1 (0.43) KDM4EALDH1A1HPGDMAPK1P2RY6
SCHEMBL4373670 0.76 P2RY6 (0.37) ADRA1DKDM4EALDH1A1CYP3A4HPGD
SCHEMBL6409879 0.75 ADRA2A (0.49) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL7572814 0.73 P2RY6 (0.33) KDM4EALDH1A1CYP3A4HPGDMAPK1
SCHEMBL21067362 0.69 PDE4B (0.46) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL6825718 0.69 RAB9A (0.46) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL4365633 0.69 SRC (0.41) MAOBCYP2D6CYP2C9CYP2C19
SCHEMBL13861954 0.68 TSHR (0.53) KDM4EALDH1A1GAAPTGS2CYP2D6
SCHEMBL25221126 0.68 SLC1A5 (0.38) KDM4EALDH1A1CYP3A4HPGDMAPK1
SCHEMBL26099141 0.68 MAPK1 (0.36) ALDH1A1MAPK1P2RY6MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874839-B1 FURAN- AND THIOPHENECARBOTHIOAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF THE REPLICATION OF HIV-1 AND HIV-1 MUTANTS UNIROYAL CHEM CO INC (US) 2002-09-18 EP disclosed
EP-0874839-A1 FURAN- AND THIOPHENECARBOTHIOAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF THE REPLICATION OF HIV-1 AND HIV-1 MUTANTS UNIROYAL CHEMICAL COMPANY, Inc. (US) 1998-11-04 EP disclosed
US-5696151-A Compounds useful for the inhibition of the replication of HIV-1 and HIV-1 mutants UNIROYAL CHEMICAL COMPANY, INC. (US) 1997-12-09 US disclosed
WO-1997019940-A1 FURAN- AND THIOPHENECARBOTHIOAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF THE REPLICATION OF HIV-1 AND HIV-1 MUTANTS UNIROYAL CHEMICAL COMPANY, INC. (US) 1997-06-05 WO disclosed