SCHEMBL758128

SCHEMBL758128

Cc1cc(Br)cnc1N1CC(C)(C)Oc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
CYP3A4 P08684 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
GAA P10253 1/20 0.34
TSHR P16473 2/20 0.33
NR3C2 P08235 1/20 0.33
AKR1B1 P15121 1/20 0.33
NPC1 O15118 2/20 0.32
MAPT P10636 2/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CASP1 P29466 1/20 0.32
CASP3 P42574 1/20 0.32
CASP4 P49662 1/20 0.32
CASP7 P55210 1/20 0.32
CASP9 P55211 1/20 0.32
CASP6 P55212 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2272405 0.80 ALDH1A1 (0.36) ALDH1A1CYP3A4TDP1MEN1KMT2A
SCHEMBL27414020 0.76 MAPT (0.42) ALDH1A1MEN1KMT2AGAANPC1
SCHEMBL27735505 0.76 NPC1 (0.32) ALDH1A1CYP3A4TDP1MEN1KMT2A
SCHEMBL756044 0.72 NR3C2 (0.60) ALDH1A1TDP1MEN1KMT2ANR3C2
SCHEMBL5140408 0.71 NR3C2 (0.41) ALDH1A1CYP3A4TDP1MEN1KMT2A
SCHEMBL9147151 0.70 CASP6 (0.38) ALDH1A1TDP1MEN1KMT2AGAA
SCHEMBL2268117 0.70 NR3C2 (0.44) ALDH1A1MEN1KMT2AGAANR3C2
SCHEMBL9146981 0.69 L3MBTL1 (0.45) ALDH1A1MEN1KMT2AGAANR3C2
Hydrochloric Acid SCHEMBL9143208 0.68 L3MBTL1 (0.44) ALDH1A1MEN1KMT2AGAANR3C2
SCHEMBL9725698 0.68 MAPT (0.42) ALDH1A1MEN1KMT2AGAAAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984345-B9 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORP (JP) 2012-03-21 EP disclosed
EP-1984345-B1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORP (JP) 2011-08-31 EP disclosed
EP-1984345-A1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS Mitsubishi Tanabe Pharma Corporation (JP) 2008-10-29 EP disclosed
WO-2007089034-A1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-08-09 WO disclosed