SCHEMBL7589926

SCHEMBL7589926

C=C1[C@@H](c2ccc(C(C)(C)C)cc2)[C@@](C)(c2ccccc2)NC(=N)N1C

nearest known ligand 0.30

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 1/20 0.30
TNKS O95271 1/20 0.30
TNKS2 Q9H2K2 1/20 0.30
PARP3 Q9Y6F1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18294767 0.91 RORC (0.31)
SCHEMBL7581116 0.88 TP53 (0.31)
SCHEMBL7589827 0.87 P2RX7 (0.34)
SCHEMBL7582511 0.86 TNKS2 (0.35) NR1H3TNKSTNKS2PARP3
SCHEMBL7579035 0.86 TNKS2 (0.35) NR1H3TNKSTNKS2PARP3
SCHEMBL13054282 0.86 TNKS2 (0.35) NR1H3TNKSTNKS2PARP3
SCHEMBL7589834 0.85 KIF11 (0.38)
SCHEMBL7589846 0.85
SCHEMBL7589861 0.81
SCHEMBL7585494 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed