SCHEMBL759272

SCHEMBL759272

CC1(C)OB(c2ccc3[nH]cc(C=O)c3c2)OC1(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C19 P33261 1/20 0.50
CYP2A6 P11509 2/20 0.44
IMPDH2 P12268 1/20 0.44
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
HASPIN Q8TF76 1/20 0.38
LPL P06858 4/20 0.36
LIPG Q9Y5X9 4/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1337551 0.80 ATM (0.41) LPLLIPGPRMT5WDR77IDO1
SCHEMBL1337645 0.79 LPL (0.42) LPLLIPGPRMT5WDR77
SCHEMBL22438423 0.76 LPL (0.38) LPLLIPGPRMT5WDR77EGFR
SCHEMBL2220082 0.75 IMPDH2 (0.44) IMPDH2CCNT1CDK9HASPINLPL
SCHEMBL1337282 0.74 LPL (0.50) LPLLIPG
SCHEMBL15617180 0.74 LIPG (0.53) IMPDH2HASPINLPLLIPGPRMT5
SCHEMBL17588945 0.74 PRMT5 (0.42) LPLLIPGPRMT5WDR77IDO1
SCHEMBL24214891 0.74 HIF1A (0.39) LIPGPRMT5WDR77CA1CA2
SCHEMBL15897087 0.74 ALDH1A1 (0.56) ALDH1A1CYP2C19KDM4EMAPTLIPG
SCHEMBL3070024 0.74 NR4A2 (0.58) MAPTPRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-8785438-B2 Imidazopyridin-2-one derivatives DAIICHI SANKYO COMPANY, LIMITED (JP) 2014-07-22 US disclosed
US-20130338156-A1 IMIDAZOPYRIDIN-2-ONE DERIVATIVES DAIICHI SANKYO COMPANY, LIMITED (JP) 2013-12-19 US disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
US-8436012-B2 Imidazopyridin-2-one derivatives DAIICHI SANKYO COMPANY, LIMITED (JP) 2013-05-07 US disclosed
US-20120053345-A1 Indazole Compounds ABBOTT LABORATORIES (US) 2012-03-01 US disclosed
US-20120053345-A1 Indazole Compounds ABBOTT LABORATORIES (US) 2012-03-01 US disclosed
EP-2308877-A1 IMIDAZOPYRIDIN-2-ON DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2011-04-13 EP disclosed
US-20110082138-A1 IMIDAZOPYRIDIN-2-ONE DERIVATIVES DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-04-07 US disclosed
EP-2303886-A2 PI3K/M TOR INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2011-04-06 EP disclosed
WO-2010008847-A2 PI3K/M TOR INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-01-21 WO disclosed
EP-2001480-A2 INDAZOLE COMPOUNDS Abbott Laboratories (US) 2008-12-17 EP disclosed
US-20070282101-A1 Indazole compounds ABBVIE INC. 2007-12-06 US disclosed
US-20070282101-A1 Indazole compounds ABBVIE INC. 2007-12-06 US disclosed
US-20070282101-A1 Indazole compounds ABBVIE INC. 2007-12-06 US disclosed
WO-2007117465-A2 INDAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2007-10-18 WO disclosed
WO-2007117465-A2 INDAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2007-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110082138-A1 IMIDAZOPYRIDIN-2-ONE DERIVATIVES MTOR, MAPKAP1, RICTOR ALDH1A1 2312/4885CYP1A2 1450/4885CYP2C19 766/4885
US-20070282101-A1 Indazole compounds CYP3A43, CYP3A7, UGT1A1 ALDH1A1 89/4885CYP1A2 15/4885CYP2C19 4/4885
US-20130338156-A1 IMIDAZOPYRIDIN-2-ONE DERIVATIVES MTOR, MAPKAP1, RICTOR ALDH1A1 2312/4885CYP1A2 1450/4885CYP2C19 766/4885
US-20120053345-A1 Indazole Compounds CYP3A43, CYP3A7, UGT1A1 ALDH1A1 89/4885CYP1A2 15/4885CYP2C19 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.