SCHEMBL7594872

SCHEMBL7594872

COc1csc(C(Cc2cc[c]c(Br)c2)C(=O)c2ccccc2)n1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 10/20 0.37
PTPN2 P17706 1/20 0.34
MRE11 P49959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7174193 0.77 PTPN1 (0.41) PTPN1PTPN2
SCHEMBL7618267 0.77 PTPN1 (0.51) PTPN1PTPN2
SCHEMBL7166523 0.76 PTPN1 (0.53) PTPN1PTPN2
SCHEMBL7183658 0.66 PLA2G4A (0.38) PTPN1PTPN2
SCHEMBL723821 0.63 CES2 (0.42)
SCHEMBL7591773 0.62 KDM4E (0.45)
SCHEMBL22344416 0.58 KDM4E (0.46)
SCHEMBL2922282 0.58 MITF (0.59) PTPN1
SCHEMBL27608960 0.58 SLC7A5 (0.61) PTPN1PTPN2
SCHEMBL3393204 0.57 L3MBTL1 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244678-A1 PHOSPHONIC ACID DERIVATIVES AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE 1B (PTP-1B) MERCK FROSST CANADA INC. (CA) 2002-10-02 EP disclosed
WO-2001046206-A1 PHOSPHONIC ACID DERIVATIVES AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE 1B (PTP-1B) MERCK FROSST CANADA & CO. (CA) 2001-06-28 WO disclosed