SCHEMBL7596015

SCHEMBL7596015

COc1cccc(CNC(=O)OC2(CCCCBr)c3ccccc3-c3ccccc32)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.48
RAB9A P51151 1/20 0.47
HPGD P15428 2/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HTT P42858 1/20 0.46
FBP1 P09467 1/20 0.46
EPHX2 P34913 2/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
NPC1 O15118 1/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43
GFER P55789 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599607 0.89 NPC1 (0.46) RAB9AHPGDLMNAALDH1A1HTT
SCHEMBL7599929 0.86 TP53 (0.39) HPGDSMN1; SMN2EPHX2MEN1GAA
SCHEMBL7600342 0.86 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2EPHX2MEN1GAA
SCHEMBL7594799 0.84 TAS1R3 (0.49) HPGDALDH1A1HTTMEN1GAA
SCHEMBL6771541 0.84 MMP13 (0.50) MMP13RAB9AHPGDLMNAALDH1A1
SCHEMBL7596021 0.81 HDAC1 (0.45) RAB9AHPGDALDH1A1HTTFBP1
SCHEMBL7596777 0.80 HTT (0.41) MMP13LMNAALDH1A1SMN1; SMN2HTT
SCHEMBL7596505 0.80 POLB (0.41) RAB9AHPGDLMNAALDH1A1SMN1; SMN2
SCHEMBL7600206 0.79 PDK2 (0.39) LMNA
SCHEMBL7599983 0.79 PDK2 (0.37) RAB9AHPGDALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255736-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) Boehringer Ingelheim Pharma KG (DE) 2002-11-13 EP disclosed
WO-2001047898-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-05 WO disclosed