Acridan

Acridan

SCHEMBL7596523

CN1c2ccccc2C(C(=O)O)c2c(-c3c(F)cccc3F)cccc21.c1ccc2c(c1)Cc1ccccc1N2

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
EGFR P00533 2/20 0.32
SRC P12931 1/20 0.32
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
KIF11 P52732 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
SLC6A2 P23975 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7796571 0.87 HDAC4 (0.46) MEN1MAPTKMT2AHDAC4HDAC7
Acridan SCHEMBL7793226 0.87 HDAC4 (0.36) MEN1MAPTKMT2AHDAC4HDAC7
Acridan SCHEMBL7755713 0.84 HDAC4 (0.36) MEN1MAPTKMT2AHDAC4HDAC7
Acridan SCHEMBL6586926 0.81 ALDH1A1 (0.32) MEN1MAPTKMT2AHDAC4HDAC7
SCHEMBL7787075 0.76 MAPT (0.39) MEN1MAPTKMT2AHDAC4HDAC7
Acridan SCHEMBL7594988 0.75 HDAC3 (0.32) HDAC4HDAC7HDAC5ALDH1A1TSHR
SCHEMBL2218310 0.73 HDAC4 (0.50) MEN1MAPTKMT2AHDAC4HDAC7
Acridan SCHEMBL7755741 0.73 HDAC4 (0.42) MEN1KMT2AHDAC4HDAC7HDAC5
SCHEMBL7787066 0.72 HDAC4 (0.44) MEN1MAPTKMT2AHDAC4HDAC7
SCHEMBL5665141 0.72 HDAC4 (0.44) MEN1MAPTKMT2AHDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778946-B1 NOVEL METHOD AND KITS FOR PRODUCING LIGHT FROM AN ACRIDAN COMPOUND LUMIGEN INC (US) 2002-10-23 EP disclosed
US-5723295-A MULTISTAGE CHEMILUMINESCENT ASSAY WITH PEROXIDASE ENZYME, PH ADJUSTMENT LUMIGEN, INC. (US) 1998-03-03 US disclosed
US-5670644-A CHEMILUMINESCENT REACTIONS, PEROXIDASE AND PH FOR IMMUNOASSAY LUMIGEN, INC. (US) 1997-09-23 US disclosed