Acridan

Acridan

SCHEMBL6586926

COc1cc(-c2c(F)ccc(F)c2F)c2c(c1)N(C)c1ccccc1C2C(=O)O.c1ccc2c(c1)Cc1ccccc1N2

nearest known ligand 0.33

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
HDAC4 P56524 2/20 0.31
HDAC7 Q8WUI4 2/20 0.31
HDAC5 Q9UQL6 2/20 0.31
PIN1 Q13526 1/20 0.31
AVPR1A P37288 6/20 0.31
BRD4 O60885 3/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
HDAC3 O15379 1/20 0.31
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7797026 0.90 HDAC4 (0.38) ALDH1A1TSHRHDAC4HDAC7HDAC5
Acridan SCHEMBL7594988 0.85 HDAC3 (0.32) ALDH1A1TSHRHDAC4HDAC7HDAC5
SCHEMBL7787075 0.83 MAPT (0.39) ALDH1A1TSHRHTR2AHTR2CHTR2B
Acridan SCHEMBL7596523 0.81 MEN1 (0.37) ALDH1A1TSHRHTR2AHTR2CHTR2B
Acridan SCHEMBL7793226 0.75 HDAC4 (0.36) ALDH1A1HDAC4HDAC7HDAC5BRD4
Acridan SCHEMBL6342017 0.74 HDAC4 (0.38) ALDH1A1TSHRHTR2AHTR2CHTR2B
Acridan SCHEMBL7755713 0.72 HDAC4 (0.36) HTR2AHTR2CHTR2BHDAC4HDAC7
SCHEMBL8877458 0.72 KDM4E (0.35) ALDH1A1TSHRHDAC4HDAC7HDAC5
SCHEMBL7797048 0.72 HDAC4 (0.39) ALDH1A1HDAC4HDAC7HDAC5PIN1
Acridan SCHEMBL7755741 0.71 HDAC4 (0.42) HTR2AHTR2CHTR2BHDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778947-B1 CHEMILUMINESCENT DETECTION OF HYDROLYTIC ENZYMES USING AN ACRIDAN LUMIGEN INC (US) 2004-05-12 EP claimed
EP-0778947-B1 CHEMILUMINESCENT DETECTION OF HYDROLYTIC ENZYMES USING AN ACRIDAN LUMIGEN INC (US) 2004-05-12 EP disclosed
US-5686258-A Chemiluminescent detection of hydrolytic enzymes using an acridan LUMIGEN, INC. (US) 1997-11-11 US disclosed