SCHEMBL7598526

SCHEMBL7598526

COc1cccc(Oc2c(OCCO)nc(C(=O)N3CCOCC3)nc2N(CC(C)C)S(=O)(=O)c2ccccc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
KEAP1 Q14145 3/20 0.40
NFE2L2 Q16236 3/20 0.40
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
EDNRA P25101 2/20 0.38
EDNRB P24530 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
NR1H2 P55055 1/20 0.37
GFER P55789 1/20 0.37
HTT P42858 2/20 0.37
MAPT P10636 2/20 0.37
PTGS2 P35354 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327772 0.81 EDNRA (0.42) KMT2AKEAP1NFE2L2SMN1; SMN2HPGD
SCHEMBL7321798 0.78 GBA1 (0.40) KMT2AALDH1A1SMN1; SMN2HPGDL3MBTL1
SCHEMBL8326904 0.77 EDNRA (0.48) EDNRAEDNRB
SCHEMBL7598517 0.75 EDNRA (0.67) EDNRAEDNRB
SCHEMBL7322839 0.73 EDNRA (0.42) KMT2AHPGDEDNRAEDNRBNR1H2
SCHEMBL8326008 0.72 EDNRA (0.47) KMT2AKEAP1NFE2L2ALDH1A1HPGD
SCHEMBL7327055 0.71 EDNRA (0.48) EDNRAEDNRB
SCHEMBL8326451 0.71 EDNRA (0.41) KMT2AALDH1A1CYP2C9HPGDEDNRA
SCHEMBL8327618 0.71 EDNRA (0.42) KMT2AEDNRAEDNRBNR1H2MAPT
SCHEMBL7330749 0.71 EDNRA (0.49) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0768304-B1 N-(Pyrimidinyl)-benzenesulfonamides as medicaments HOFFMANN LA ROCHE (CH) 2002-05-22 EP disclosed