SCHEMBL7599531

SCHEMBL7599531

Cc1cc(Cl)cc(Cl)c1CNc1c(NC(C)(C)C)c(=O)c1=O

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
P2RX7 Q99572 17/20 0.39
RAPGEF4 Q8WZA2 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7895615 0.89 L3MBTL1 (0.39) ALDH1A1HPGDSMN1; SMN2RAPGEF4EPHX2
SCHEMBL4261100 0.88 ALDH1A1 (0.42) ALDH1A1HPGDSMN1; SMN2P2RX7RAPGEF4
SCHEMBL7602216 0.82 ALDH1A1 (0.41) ALDH1A1HPGDSMN1; SMN2P2RX7
SCHEMBL7599406 0.82 ALDH1A1 (0.41) ALDH1A1HPGDSMN1; SMN2P2RX7
SCHEMBL7597275 0.82 ALDH1A1 (0.41) ALDH1A1HPGDSMN1; SMN2P2RX7
SCHEMBL7894120 0.81 CHEK2 (0.33) P2RX7RAPGEF4
SCHEMBL7895056 0.81 CYP3A4 (0.41) HPGDP2RX7
SCHEMBL7597337 0.80 ALDH1A1 (0.42) ALDH1A1HPGDSMN1; SMN2P2RX7EPHX2
SCHEMBL7597876 0.80 ALDH1A1 (0.40) ALDH1A1HPGDSMN1; SMN2P2RX7EPHX2
SCHEMBL7895628 0.78 ROCK2 (0.32) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934257-B1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES WYETH CORP (US) 2002-12-11 EP claimed
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP claimed
EP-0934257-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1999-08-11 EP claimed
US-5763474-A SMOOTH MUSCLE RELAXANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-06-09 US claimed
WO-1998002413-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1998-01-22 WO claimed
EP-0934257-B1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES WYETH CORP (US) 2002-12-11 EP disclosed
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP disclosed
EP-0934257-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1999-08-11 EP disclosed
US-5763474-A SMOOTH MUSCLE RELAXANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-06-09 US disclosed
WO-1998002413-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1998-01-22 WO disclosed