SCHEMBL7600972

SCHEMBL7600972

O=C(O)C[C@H](c1ccc2[nH]c(=O)oc2c1)N1CCN(CCCC2=CC=C3CCCNC3N2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 13/20 0.44
ITGB3 P05106 11/20 0.44
ITGB8 P26012 6/20 0.40
ITGB6 P18564 5/20 0.40
ITGA5 P08648 4/20 0.39
ITGB1 P05556 1/20 0.39
ITGA2B P08514 1/20 0.39
HTR1A P08908 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
GRIN2B Q13224 1/20 0.32
ENPP2 Q13822 1/20 0.30
ATXN2 Q99700 1/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7596629 1.00 ITGAV (0.44) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL4374388 0.85 ITGB3 (0.45) ITGAVITGB3GRIN2BENPP2ATXN2
SCHEMBL7595642 0.84 ITGAV (0.63) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7553084 0.84 ITGAV (0.63) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7592559 0.84 ITGAV (0.63) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7559347 0.83 ITGAV (0.49) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7584472 0.82 ITGAV (0.47) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7597852 0.82 ITGAV (0.47) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7596086 0.82 ITGAV (0.47) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7592874 0.82 ITGAV (0.42) ITGAVITGB3ITGB8ITGB6ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-10-04 EP disclosed
WO-1999031099-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed