SCHEMBL7601343

SCHEMBL7601343

FC(F)(F)c1ccccc1OCCN1CCNCC1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.60
HTR2A P28223 2/20 0.60
DRD2 P14416 5/20 0.59
LTA4H P09960 2/20 0.59
PTGS2 P35354 1/20 0.59
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C19 P33261 1/20 0.56
HSD17B10 Q99714 1/20 0.56
HTR1A P08908 1/20 0.55
HTR7 P34969 1/20 0.55
KCNH2 Q12809 1/20 0.50
ALDH1A1 P00352 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
KDM4E B2RXH2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14970707 0.85 LTA4H (0.73) DRD2LTA4HPTGS2CYP1A2CYP2D6
SCHEMBL17848348 0.85 LTA4H (0.73) DRD2LTA4HPTGS2CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL14969001 0.84 LTA4H (0.71) DRD2LTA4HPTGS2CYP1A2CYP2D6
SCHEMBL17848474 0.82 DRD2 (0.58) HTR2CHTR2ADRD2LTA4HPTGS2
SCHEMBL17848431 0.82 DRD2 (0.61) HTR2CHTR2ADRD2LTA4HPTGS2
SCHEMBL2158197 0.81 KDM4E (0.60) HTR2CLTA4HCYP1A2CYP2D6CYP2C19
SCHEMBL17848636 0.81 HTR7 (0.61) HTR2ADRD2LTA4HPTGS2CYP1A2
SCHEMBL17848618 0.81 HTR1A (0.61) HTR2CHTR2ADRD2LTA4HPTGS2
SCHEMBL17848384 0.79 DRD2 (0.71) DRD2LTA4HPTGS2CYP1A2CYP2D6
SCHEMBL28311407 0.78 TSHR (0.72) HTR2CHTR2ALTA4HCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246820-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2002-10-09 EP disclosed
WO-2001049683-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2001-07-12 WO disclosed