SCHEMBL7604082

SCHEMBL7604082

NC(=O)c1ccc(C(CC2(c3ccc(Cl)cc3)CCC2)C2CCCNC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.35
CHEK1 O14757 7/20 0.35
CDK2AP1 O14519 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7558108 0.72 SLC6A4 (0.37) SLC6A2SLC6A4SLC6A3
SCHEMBL4475880 0.68 HSD11B1 (0.41) HSD11B1CHEK1KCNH2
SCHEMBL3432643 0.65 OPRD1 (0.45) CHEK1SLC6A2SLC6A4SLC6A3
SCHEMBL6508980 0.65 KMT2A (0.48) CHEK1CDK2AP1SLC6A4SLC6A3
SCHEMBL3299919 0.64 SLC6A4 (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL3297642 0.64 SLC6A4 (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL3297878 0.64 SLC6A4 (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL3297637 0.64 SLC6A4 (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL4671412 0.63 MGLL (0.49)
SCHEMBL7354541 0.63 OPRM1 (0.41) CHEK1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002069895-A2 HETEROCYCLIC ANALGESIC COMPOUNDS AND METHODS OF USE THEREOF SEPRACOR, INC. (US) 2002-09-12 WO disclosed