SCHEMBL7604548

SCHEMBL7604548

CCC[C@H](NC(=O)C(CCN1C(=O)N(C)C(C)(C)C1=O)SC(C)=O)C(=O)N[C@H](C(=O)NC)C(C)(C)C

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 18/20 0.63
MMP1 P03956 16/20 0.63
MMP2 P08253 13/20 0.63
MMP9 P14780 8/20 0.63
MMP7 P09237 5/20 0.63
MMP13 P45452 4/20 0.63
MMP14 P50281 1/20 0.63
MMP8 P22894 1/20 0.49
ADAM17 P78536 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606336 0.91 MMP1 (0.77) MMP3MMP1MMP2MMP9MMP7
SCHEMBL6760102 0.88 MMP3 (0.81) MMP3MMP1MMP2MMP9MMP7
SCHEMBL6555661 0.82 MMP1 (0.78) MMP3MMP1MMP2MMP9MMP7
SCHEMBL6554365 0.79 MMP2 (0.67) MMP3MMP1MMP2MMP9MMP7
SCHEMBL14156438 0.79 MMP1 (0.67) MMP3MMP1MMP2MMP9MMP7
SCHEMBL6766456 0.79 MMP1 (0.67) MMP3MMP1MMP2MMP9MMP7
SCHEMBL8535220 0.78 MMP1 (0.48) MMP3MMP1MMP2MMP9MMP7
Rebimastat SCHEMBL12247619 0.77 MMP1 (1.00) MMP3MMP1MMP2MMP9MMP7
Rebimastat SCHEMBL12946005 0.77 MMP1 (1.00) MMP3MMP1MMP2MMP9MMP7
Rebimastat SCHEMBL645121 0.77 MMP1 (1.00) MMP3MMP1MMP2MMP9MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859784-B1 THIO-SUBSTITUTED PEPTIDES AS INHIBITORS FOR METALLOPROTEINASES AND TNF LIBERATION DARWIN DISCOVERY LTD (GB) 2002-12-18 EP disclosed
US-5981490-A ADMINISTERING A PEPTIDYL COMPOUND FOR TREATMENT IN A HUMAN OR ANIMAL OF A CONDITION ASSOCIATED WITH MATRIX METALIOPROTEINASES OR THAT IS MEDIATED BY TUMOR NECROSIS FACTOR ALPHA OR L-SELECTIN SHEDDASE DARWIN DISCOVERY, LTD. (GB) 1999-11-09 US disclosed