SCHEMBL7605822

SCHEMBL7605822

O=C(N[C@@H](Cc1ccc(CC(O)c2c(Cl)cccc2Cl)cc1)C(=O)O)c1cccnc1Cl

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.59
ITGA4 P13612 14/20 0.59
ITGB2 P05107 1/20 0.54
ICAM1 P05362 1/20 0.54
ITGAL P20701 1/20 0.54
ITGB7 P26010 3/20 0.54
ITGA5 P08648 5/20 0.48
ITGB3 P05106 2/20 0.47
ITGAV P06756 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7605825 1.00 ITGB1 (0.59) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7605742 0.87 ITGB1 (0.50) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7613198 0.84 ITGB1 (0.59) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7607529 0.83 ITGA4 (0.59) ITGB1ITGA4ITGA5ITGB3ITGAV
SCHEMBL7607510 0.83 ITGB1 (0.58) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7607515 0.83 ITGB1 (0.58) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7991508 0.83 ITGB1 (0.59) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7606675 0.79 ITGB1 (0.55) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL7709504 0.78 ITGB1 (0.55) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4625285 0.78 ITGB1 (0.75) ITGB1ITGA4ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020035127-A1 Phenylalanine derivatives CELLTECH THERAPEUTIS, LIMITED 2002-03-21 US disclosed
US-6329372-B1 HETEROCYCLIC AMIDE COMPOUNDS ARE ABLE TO INHIBIT THE BINDING OF ALPHA4 INTEGRINS TO THEIR LIGANDS AND ARE OF USE IN THE PROPHYLAXIS AND TREATMENT OF IMMUNE OR INFLAMMATORY DISORDERS. CELLTECH THERAPEUTICS LIMITED (GB) 2001-12-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020035127-A1 Phenylalanine derivatives PAH, VCAM1, IL4I1 ITGB1 8/4885ITGA4 5/4885ITGB2 23/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.